Zaldaride maleate, MedChemExpress

MedChemExpress Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride maleate (CGS-9343B) inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM. Zaldaride maleate (CGS-9343B) prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR.

Brand:  Medchem Express HY-105118A

Product Code. 16486727

Description

Zaldaride maleate (CGS-9343B) is a potent, orally active and selective inhibitor of calmodulin. Zaldaride maleate (CGS-9343B) inhibits CaM (calmodulin)-stimulated cAMP phosphodiesterase activity, with an IC50 of 3.3 nM. Zaldaride maleate (CGS-9343B) prevents estrogen-induced transcription activation by ER, reversibly blocks voltage-activated Na+, Ca2+ and K+ currents in PC12 cells and inhibits nAChR.

Specifications

• Chemical Name or Material: Zaldaride maleate
• Color: White
• Molecular Formula: C₃₀H₃₂N₄O₆
• Synonym: CGS-9343B KW 5617
• Molecular Weight (g/mol): 544.6
• Percent Purity: 98.0%
• Physical Form: Solid

• CAS: 109826-27-9
• Purity Grade Notes: Research
• Quantity: 5 mg
• SMILES: O=C(O)/C=C\C(O)=O.CC1(C2=CC=CN2C3=CC=CC=C3CO1)CN4CCC(N5C6=C(C=CC=C6)NC5=O)CC4
• Formula Weight: 544.6
• Grade: Research
• For Use With (Application): Neuroscience-Neuromodulation

Research purposes only