Trimipramine maleate, MedChemExpress

Product Code. 16468686

Brand: Medchem Express HYB1213

Description

MedChemExpress Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively.

Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine maleate has vascular activity and anxiolytic efficacy.

Specifications

• Chemical Name or Material: Trimipramine maleate
• CAS: 521-78-8
• Color: White
• Purity Grade Notes: Research
• Molecular Formula: C₂₄H₃₀N₂O₄
• Quantity: 100 mg
• Solubility Information: DMSO : ≥ 100 mg/mL (243.60 mM) ∣H2O : 14.29 mg/mL (34.81 mM; ultrasonic and warming and heat to 60°C)
• SMILES: CC(CN(C)C)CN1C2=C(C=CC=C2)CCC3=C1C=CC=C3.O=C(O)/C=C\C(O)=O
• Molecular Weight (g/mol): 410.51
• Formula Weight: 410.51
• Percent Purity: 99.97%
• Grade: Research
• Physical Form: Solid
• For Use With (Application): Neuroscience-Neuromodulation

Research purposes only