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RPR-260243, MedChemExpress

Product Code. 16487208
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Quantity:
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10 mg
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50mg
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Product Code. 16487208

Brand: Medchem Express HY16915

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Description

MedChemExpress RPR-260243, a potent activator of human ether-a-go-go-related gene (hERG), slows deactivation and attenuates inactivation of hERG1 channels. RPR260243-modified HERG currents are inhibited by Dofetilide (IC50=58 nM). RPR260243 displays no activator-like effects on other voltage-dependent ion channels, including the closely related ERG3 K+ channel.

RPR-260243, a potent activator of human ether-a-go-go-related gene (hERG), slows deactivation and attenuates inactivation of hERG1 channels. RPR260243-modified HERG currents are inhibited by Dofetilide (IC50=58 nM). RPR260243 displays no activator-like effects on other voltage-dependent ion channels, including the closely related ERG3 K+ channel.

Specifications

Chemical Name or Material RPR-260243
CAS 668463-35-2
Color Light Brown
Purity Grade Notes Research
Molecular Formula C28H25F3N2O4
Quantity 10 mg
Solubility Information DMSO : 10 mg/mL (19.59 mM; Need ultrasonic)
SMILES O=C([C@H]1CN(CC#CC2=CC(F)=CC(F)=C2F)CC[C@H]1CCC(C3=CC=NC4=CC=C(OC)C=C34)=O)O
Molecular Weight (g/mol) 510.5
Formula Weight 510.5
Percent Purity 98.84%
Grade Research
Physical Form Solid
For Use With (Application) COVID-19-immunoregulation
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Research purposes only

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