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Tocris Bioscience™ R 59-022

Diacylglycerol kinase inhibitor; increases PKC activity

POA

Specifications

Purity >98%
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Description

Description

Diacylglycerol (DAG) kinase inhibitor (IC50 = 2.8 μM); increases protein kinase C activity. Potentiates thrombin-induced platelet aggregation and induces neutrophil chemotaxis. Inhibits U46619-induced contractions in mouse aorta and porcine coronary artery.
Specifications

Specifications

>98%
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