Omipalisib, MedChemExpress

MedChemExpress Omipalisib (GSK2126458) is an orally active and highly selective inhibitor of PI3K with Kis of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2, respectively. Omipalisib has anti-cancer activity.

Product Code	Brand	Quantity
16456487	Medchem Express HY-10297	5 mg
16430147	Medchem Express HY-10297	50 mg
16403768	Medchem Express HY-10297	10 mg

Description

Omipalisib (GSK2126458) is an orally active and highly selective inhibitor of PI3K with Kis of 0.019 nM/0.13 nM/0.024 nM/0.06 nM and 0.18 nM/0.3 nM for p110α/β/δ/γ, mTORC1/2, respectively. Omipalisib has anti-cancer activity.

Specifications

• Chemical Name or Material: Omipalisib
• Color: Light Yellow
• Molecular Formula: C₂₅H₁₇F₂N₅O₃S
• Solubility Information: DMSO : 50 mg/mL (98.91 mM; Need ultrasonic)
• Molecular Weight (g/mol): 505.5
• Percent Purity: 96.89%
• Physical Form: Solid

• CAS: 1086062-66-9
• Purity Grade Notes: Research
• Synonym: GSK2126458 GSK458
• SMILES: COC1=NC=C(C=C1NS(C2=CC=C(C=C2F)F)(=O)=O)C3=CC=C(C4=C3)N=CC=C4C5=CN=NC=C5
• Formula Weight: 505.5
• Grade: Research
• For Use With (Application): Cancer-Kinase/protease

Safety and Handling

missing translation for 'shelfLife' : Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month

Recommended Storage : Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month

Research purposes only