Lumateperone tosylate, MedChemExpress

Product Code. 16440338

Brand: Medchem Express HY19733

Description

MedChemExpress Lumateperone (ITI-007) tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia.

Lumateperone (ITI-007) tosylate is a 5-HT2A receptor antagonist (Ki = 0.54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator. Lumateperone tosylate has anticancer activity and can also be used in studies of psychiatric disorders such as schizophrenia.

Specifications

• Chemical Name or Material: Lumateperone tosylate
• CAS: 1187020-80-9
• Color: Gray
• Purity Grade Notes: Research
• Molecular Formula: C₃₁H₃₆FN₃O₄S
• Quantity: 5 mg
• Synonym: ITI-007 tosylate
• Solubility Information: DMSO : 100 mg/mL (176.77 mM; Need ultrasonic) ∣H2O : 1 mg/mL (1.77 mM; ultrasonic and warming and heat to 80°C)
• SMILES: O=C(C1=CC=C(F)C=C1)CCCN2CC[C@@](N3CCN(C)C4=C3C5=CC=C4)([H])[C@@]5([H])C2.O=S(C6=CC=C(C)C=C6)(O)=O
• Molecular Weight (g/mol): 565.7
• Formula Weight: 565.7
• Percent Purity: 96.56%
• Grade: Research
• Physical Form: Solid
• For Use With (Application): Neuroscience-Neuromodulation

Research purposes only