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GSK1904529A, MedChemExpress

Product Code. 16480377
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Product Code. 16480377

Brand: Medchem Express HY10524

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Description

MedChemExpress GSK1904529A is a potent, selective, orally active, and ATP-competitive inhibitor of insulin-like growth factor-1 receptor (IGF-1R) and insulin receptor (IR), with IC50s of 27 and 25 nM, respectively. GSK1904529A shows poor activity (IC50>1 μM) in 45 other serine/threonine and tyrosine kinases. GSK1904529A exhibits anti-tumor activity.

GSK1904529A is a potent, selective, orally active, and ATP-competitive inhibitor of insulin-like growth factor-1 receptor (IGF-1R) and insulin receptor (IR), with IC50s of 27 and 25 nM, respectively. GSK1904529A shows poor activity (IC50>1 μM) in 45 other serine/threonine and tyrosine kinases. GSK1904529A exhibits anti-tumor activity.

Specifications

Chemical Name or Material GSK1904529A
CAS 1089283-49-7
Color Yellow
Purity Grade Notes Research
Molecular Formula C44H47F2N9O5S
Quantity 50 mg
Solubility Information DMSO : 50 mg/mL (58.69 mM; Need ultrasonic)
SMILES O=C(C1=CC(C2=C(N3C=CC=CC3=N2)C4=NC(NC5=CC(CC)=C(C=C5OC)N6CCC(CC6)N7CCN(CC7)S(=O)(C)=O)=NC=C4)=CC=C1OC)NC8=C(C=CC=C8F)F
Molecular Weight (g/mol) 851.96
Formula Weight 851.96
Percent Purity 99.66%
Grade Research
Physical Form Solid
For Use With (Application) Cancer-Kinase/protease
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Research purposes only

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