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Grapiprant, MedChemExpress

Product Code. 16499717
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Product Code. 16499717

Brand: Medchem Express HY16781

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Description

MedChemExpress Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2). Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor with IC50 value of 35 nM and Ki value of 24 nM. Grapiprant has the potential for osteoarthritic pain and inflammation treatment[3] .

Grapiprant (CJ-023423) is a selective EP4 receptor antagonist whose physiological ligand is prostaglandin E2 (PGE2). Grapiprant displaces [3H]-PGE2 (1 nM) binding to dog recombinant EP4 receptor with IC50 value of 35 nM and Ki value of 24 nM. Grapiprant has the potential for osteoarthritic pain and inflammation treatment[3] .

Specifications

Chemical Name or Material Grapiprant
CAS 415903-37-6
Color Off-White
Purity Grade Notes Research
Molecular Formula C26H29N5O3S
Quantity 5 mg
Synonym CJ-023423 RQ-00000007 AAT-007
Solubility Information DMSO : ≥ 50 mg/mL (101.71 mM)
SMILES O=S(C1=CC=C(C)C=C1)(NC(NCCC2=CC=C(N3C(CC)=NC4=C3C=C(C)N=C4C)C=C2)=O)=O
Molecular Weight (g/mol) 491.61
Formula Weight 491.61
Percent Purity 99.02%
Grade Research
Physical Form Solid
For Use With (Application) Metabolism-protein/nucleotide metabolism
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Research purposes only

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