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GR 125487 sulfamate, Tocris Bioscience™

£209.16 - £797.91

CAS	859502-43-5
Molecular Formula	C19H29FN4O8S2
Molecular Weight (g/mol)	524.579
InChI Key	VQJFDBXITIOGJM-UHFFFAOYSA-N
Synonym	gr 125487 sulfamate, gr 125487 sulfamate salt, 5-fluoro-2-methoxy-1-2-methylsulfonyl amino ethyl-4-piperidinyl-1h-indole-3-methylcarboxylate sulfamate, tocris-1658, gr-125487 sulfamate salt, 1-2-methanesulfonamido ethyl piperidin-4-yl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate; sulfamic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 5-fluoro-2-methoxy-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, sulfamate 1:1
PubChem CID	6604955
IUPAC Name	[1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate;sulfamic acid
SMILES	COC1=C(C2=C(N1)C=CC(=C2)F)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C.NS(=O)(=O)O

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Product Code	Brand	Quantity	Price	Quantity & Availability
Product Code	Brand	Quantity	Price	Quantity & Availability
18065422 View Documents Promotion Details missing translation for 'viewProductCertificates'	Tocris Bioscience 1658/10	10 mg	£209.16 10mg View alternative products Save Up to »		Please sign in to purchase this item. Need a web account? Register with us today!

18055002 View Documents Promotion Details missing translation for 'viewProductCertificates'	Tocris Bioscience 1658/50	50 mg	£797.91 50mg View alternative products Save Up to »		Please sign in to purchase this item. Need a web account? Register with us today!

Description

Potent and selective 5-HT4 receptor antagonist (Ki = 0.19 nM for porcine 5-HT4). Centrally active following systemic administration in vivo.

Specifications

Chemical Identifiers

CAS	859502-43-5
Molecular Weight (g/mol)	524.579
Synonym	gr 125487 sulfamate, gr 125487 sulfamate salt, 5-fluoro-2-methoxy-1-2-methylsulfonyl amino ethyl-4-piperidinyl-1h-indole-3-methylcarboxylate sulfamate, tocris-1658, gr-125487 sulfamate salt, 1-2-methanesulfonamido ethyl piperidin-4-yl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate; sulfamic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 5-fluoro-2-methoxy-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, sulfamate 1:1
IUPAC Name	[1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate;sulfamic acid

Molecular Formula	C19H29FN4O8S2
InChI Key	VQJFDBXITIOGJM-UHFFFAOYSA-N
PubChem CID	6604955
SMILES	COC1=C(C2=C(N1)C=CC(=C2)F)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C.NS(=O)(=O)O

CAS	859502-43-5
Synonym	gr 125487 sulfamate, gr 125487 sulfamate salt, 5-fluoro-2-methoxy-1-2-methylsulfonyl amino ethyl-4-piperidinyl-1h-indole-3-methylcarboxylate sulfamate, tocris-1658, gr-125487 sulfamate salt, 1-2-methanesulfonamido ethyl piperidin-4-yl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate; sulfamic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl 5-fluoro-2-methoxy-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 5-fluoro-2-methoxy-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, sulfamate 1:1
SMILES	COC1=C(C2=C(N1)C=CC(=C2)F)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C.NS(=O)(=O)O
Molecular Weight (g/mol)	524.579
Formula Weight	524.58
Chemical Name or Material	GR 125487 sulfamate

Molecular Formula	C19H29FN4O8S2
InChI Key	VQJFDBXITIOGJM-UHFFFAOYSA-N
IUPAC Name	[1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 5-fluoro-2-methoxy-1H-indole-3-carboxylate;sulfamic acid
PubChem CID	6604955
Percent Purity	>98%

Safety and Handling

Recommended Storage : Desiccate at Room Temperature