Glutaminase-IN-1, MedChemExpress

Product Code. 16441077

Brand: Medchem Express HY114334

Description

MedChemExpress Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.

Glutaminase-IN-1 (CB839 derivative), a CB839 derivative, is an allosteric inhibitor of 1,3,4-selenadiazole-containing kidney-type glutaminase (KGA), with an IC50 of 1 nM. Glutaminase-IN-1 (CB839 derivative) shows improved cellular uptake and antitumor activity.

Especificaciones

• Chemical Name or Material: Glutaminase-IN-1
• CAS: 2247127-79-1
• Color: Yellow
• Purity Grade Notes: Research
• Molecular Formula: C₂₆H₂₄F₃N₇O₃Se
• Quantity: 50 mg
• Synonym: CB839 derivative
• Solubility Information: DMSO : 125 mg/mL (202.11 mM; Need ultrasonic) ∣H2O : < 0.1 mg/mL (insoluble)
• SMILES: O=C(NC1=NN=C(CCCCC2=NN=C(NC(CC3=CC=CC(OC(F)(F)F)=C3)=O)C=C2)[Se]1)CC4=NC=CC=C4
• Molecular Weight (g/mol): 618.47
• Formula Weight: 618.47
• Percent Purity: 98.65%
• Grade: Research
• Physical Form: Solid
• For Use With (Application): Cancer-programmed cell death

Research purposes only