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Tocris Bioscience™ CMPD101
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Product Code. 18744519
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10 mg
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10mg
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Product Code. 18744519 Supplier Tocris Bioscience™ Supplier No. 5642/10

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Description

Potent and selective GRK2/3 inhibitor

CMPD101 is a potent and selective GRK2/3 inhibitor (IC50 values are 32 and 54 nM for GRK3 and GRK2, respectively). Exhibits selectivity for GRK2/3 over GRK1/5. Reduces DAMGO -induced desensitization and internalization of μ-opioid receptors.
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Specifications

Chemical Name or Material 3-[[[4-Methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide
CAS 865608-11-3
Quantity 10 mg
Target G Protein (Heterotrimeric) Inhibitors
Molecular Formula C24H21F3N6O
Formula Weight 466.46
Purity >98%
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