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Aprocitentan, MedChemExpress

Product Code. 16499437
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Product Code. 16499437

Brand: Medchem Express HY15895

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Description

MedChemExpress Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.

Aprocitentan (ACT-132577) is the major and pharmacologically active metabolite of Macitentan. Aprocitentan is dual ETA/ETB antagonist with IC50s of 3.4 nM and 987 nM, and pA2 valus of 6.7 and 5.5, respectively.

Specifications

Chemical Name or Material Aprocitentan
CAS 1103522-45-7
Color White
Purity Grade Notes Research
Molecular Formula C16H14Br2N6O4S
Quantity 5 mg
Synonym ACT-132577
Solubility Information DMSO : ≥ 46 mg/mL (84.22 mM)
SMILES O=S(N)(NC1=NC=NC(OCCOC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)=O
Molecular Weight (g/mol) 546.19
Formula Weight 546.19
Percent Purity 98.03%
Grade Research
Physical Form Solid
For Use With (Application) COVID-19-immunoregulation
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Research purposes only

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