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A-381393, MedChemExpress

Product Code. 16471117
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Product Code. 16471117

Brand: Medchem Express HY116941

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Description

MedChemExpress A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM).

A-381393 is a potent, selective, brain penetrate dopamine D4 receptor antagonist, with Kis of 1.5, 1.9 and 1.6 nM for human dopamine D4.4, D4.2, and D4.7 receptor, respectively, >2700-fold selectivity over D1, D2, D3 and D5 dopamine receptors. A-381393 shows moderate affinity for 5-HT2A (Ki, 370 nM).

Specifications

Chemical Name or Material A-381393
Physical Form Solid
CAS 726174-00-1
Color Light Yellow
Quantity 50 mg
Purity Grade Notes Research
Molecular Formula C20H24N4
For Use With (Application) Neuroscience-Neuromodulation
Solubility Information DMSO : 51.67 mg/mL (161.25 mM; Need ultrasonic)
SMILES CC1=CC=C(C=C1C)N2CCN(CC2)CC3=NC4=CC=CC=C4N3
Molecular Weight (g/mol) 320.43
Formula Weight 320.43
Percent Purity 99.9%
Grade Research
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Research purposes only

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