1A-116, MedChemExpress

Product Code. 16442926

Brand: Medchem Express HY104064

Description

MedChemExpress 1A-116, a potent Rac1 inhibitor, is specific for W56 residues, can prevent EGF-induced Rac1 activation and block Rac1-P-Rex1 interaction. 1A-116 can induce apoptosis and inhibit cell proliferation, migration and cycle progression in a concentration-dependent manner. 1A-116 also demonstrates a high antimetastatic activity in vivo.

1A-116, a potent Rac1 inhibitor, is specific for W56 residues, can prevent EGF-induced Rac1 activation and block Rac1-P-Rex1 interaction. 1A-116 can induce apoptosis and inhibit cell proliferation, migration and cycle progression in a concentration-dependent manner. 1A-116 also demonstrates a high antimetastatic activity in vivo.

Specifications

• Chemical Name or Material: 1A-116
• Physical Form: Solid
• CAS: 1430208-73-3
• Color: Off-White
• Quantity: 25 mg
• Purity Grade Notes: Research
• Molecular Formula: C₁₆H₁₆F₃N₃
• For Use With (Application): Cancer-Kinase/protease
• Solubility Information: DMSO : 100 mg/mL (325.40 mM; Need ultrasonic)
• SMILES: N=C(NC1=CC=CC=C1C(F)(F)F)NC2=CC(C)=CC(C)=C2
• Molecular Weight (g/mol): 307.31
• Formula Weight: 307.31
• Percent Purity: 99.39%
• Grade: Research

Research purposes only