CAS RN 1221186-53-3

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Tocris Bioscience™ TEPP 46

Potent and selective pyruvate kinase M2 (PKM2) allosteric activator

Pricing and Availability
Specifications

Target	PKM2
CAS	1221186-53-3
Purity	0.98
Chemical Name or Material	6-[(3-Aminophenyl)methyl]-4,6-dihydro-4-methyl-2-(methylsulfinyl)-5H-thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one
Recommended Storage	Store at -20°C
Molecular Formula	C₁₇H₁₆N₄O₂S₂

TEPP-46, MedChemExpress

MedChemExpress TEPP-46 (ML-265) is a potent and selective pyruvate kinase M2 (PKM2) activator with an AC50 of 92 nM, showing little or no effect on PKM1, PKL and PKR.

Pricing and Availability
Specifications

Molecular Weight (g/mol)	372.46
Color	Light Yellow
Physical Form	Solid
Chemical Name or Material	TEPP-46
Grade	Research
SMILES	O=C1C(N(C)C2=C3SC(S(C)=O)=C2)=C3C=NN1CC4=CC=CC(N)=C4
For Use With (Application)	Cancer-Kinase/protease
Percent Purity	95.86%
CAS	1221186-53-3
Solubility Information	DMSO : 50 mg/mL (134.24 mM; Need ultrasonic)
Synonym	ML-265
Purity Grade Notes	Research
Recommended Storage	Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month
Shelf Life	Powder -20°C 3 years, 4°C 2 years∣In solvent -80°C 6 months, -20°C 1 month
Molecular Formula	C₁₇H₁₆N₄O₂S₂
Formula Weight	372.46

CAS RN 1221186-53-3

CAS RN 1221186-53-3

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