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Tocris Bioscience™ UBP 310

GluK1-selective kainate antagonist

Brand:  Tocris Bioscience™ 362110

Code : Z1

Additional Details : Weight : 0.00001kg

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Product Code. 13443304

  • £155.76 / 10mg

Estimated Shipment date
from Supplier 29-08-2019

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Description

Description

GluK1 (formerly GLUK5) kainate receptor antagonist (IC50 = 130 nM); also blocks recombinant homomeric GluK3 (forrmerly GLUK7) receptors. Displays 12,700-fold selectivity for GluK1 (formerly GLUK5) over GluK2 (formerly GLUK6). Exhibits no activity at mGlu group I or NMDA receptors at concentrations of up to 10 μM. Apparent KD value is 18 ± 4 nM for depression of kainate responses on the dorsal root.

Please refer to IUPHAR Guide to Pharmacology for the most recent naming conventions.

Specifications

Specifications

UBP 310
>98
10mg
UBP 310
353.35
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