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Tocris Bioscience™ TY 52156

S1P3 receptor antagonist

POA

Specifications

Product Type TY 52156
Description TY 52156
Molecular Weight (g/mol) 364.27
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Description

Description

S1P3 receptor antagonist (Ki = 110 nM); inhibits S1P-induced Ca2+ release in HUVEC cells. Suppresses FTY-720-induced S1P3 receptor-mediated bradycardia in vivo. Also inhibits S1P-induced breast cancer stem cell expansion in vitro. Orally bioavailable.
Specifications

Specifications

TY 52156
TY 52156
364.27
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