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Thioperamide, Tocris Bioscience™

H3 antagonist; also H4 inverse agonist

Brand:  Tocris (Bio-Techne) 0644/10

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 10mg

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Product Code. 13437843

  • £114.75 / 10mg

Estimated Shipment
28-06-2019

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Description

Description

Potent histamine H3 and H4 antagonist/inverse agonist. Ki values are 25 and 27 nM for human recombinant H3 and H4 receptors respectively. Blocks eosinophil shape change (IC50 = 1.4 μM) and chemotaxis (IC50 = 519 nM) induced by histamine. Freely crosses the blood-brain barrier. Also available as part of the Histamine H3 Receptor Tocriset™ .
Specifications

Chemical Identifiers

106243-16-7
408.517
1-piperidinecarbothioamide, n-cyclohexyl-4-1h-imidazol-4-yl-, 2z-2-butenedioate 1:1
but-2-enedioic acid;N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
C19H28N4O4S
WUYMIKDBRCCYGE-UHFFFAOYSA-N
53393972
C1CCC(CC1)NC(=S)N2CCC(CC2)C3=CN=CN3.C(=CC(=O)O)C(=O)O

Specifications

Thioperamide
106243-16-7
1-piperidinecarbothioamide, n-cyclohexyl-4-1h-imidazol-4-yl-, 2z-2-butenedioate 1:1
C1CCC(CC1)NC(=S)N2CCC(CC2)C3=CN=CN3.C(=CC(=O)O)C(=O)O
408.517
292.44
10mg
C19H28N4O4S
WUYMIKDBRCCYGE-UHFFFAOYSA-N
but-2-enedioic acid;N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
53393972
>99%
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