SB 366791, Tocris Bioscience™
Potent, selective, competitive TRPV1 antagonist
Brand: Tocris (Bio-Techne) 161550
Code : Z1
Additional Details : Weight : 0.01000kg
DescriptionPotent, selective and competitive vanilloid TRPV1 receptor antagonist (pA2 = 7.71 at hVR1); antagonizes hTRPV1 receptors activated by agonists, noxious heat, but not protons. Displays selectivity over a wide range of receptors and systems including CB1 and CB2 receptors, voltage-gated Ca2+ channels and the hyperpolarization-activated current (Ih). Also available as part of the Vanilloid TRPV1 Receptor Tocriset™ .