missing translation for 'onlineSavingsMsg'
Learn More

SB 243213 dihydrochloride, Tocris Bioscience™

Selective 5-HT2C inverse agonist

Brand:  RD Systems (Bio-Techne) 3527/10

Code : Z1

Additional Details : Weight : 0.00010kg

Quantity 10mg

 View more versions of this product

Product Code. 13463134

  • £191.40 / 10mg


Estimated Shipment
03-12-2018
Add to basket

Description

Description

Selective 5-HT2C inverse agonist (pKb = 9.8). Displays selectivity over other 5-HT2 subtypes (pKi values are 6.8, 7.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C respectively); also exhibits >100-fold selectivity over 50 other receptors, ion channels and enzymes. Displays anxiolytic activity in rat models.
Specifications

Chemical Identifiers

200940-23-4
501.331
sb 243213 dihydrochloride, 2,3-dihydro-5-methyl-n-6-2-methyl-3-pyridinyl oxy-3-pyridinyl-6-trifluoromethyl-1h-indole-1-carboxamide dihydrochloride
5-methyl-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide;dihydrochloride
C22H21Cl2F3N4O2
UKMTYUXWLKQDNT-UHFFFAOYSA-N
90488853
CC1=C(C=C2C(=C1)CCN2C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C)C(F)(F)F.Cl.Cl

Specifications

SB 243213 dihydrochloride
200940-23-4
sb 243213 dihydrochloride, 2,3-dihydro-5-methyl-n-6-2-methyl-3-pyridinyl oxy-3-pyridinyl-6-trifluoromethyl-1h-indole-1-carboxamide dihydrochloride
CC1=C(C=C2C(=C1)CCN2C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C)C(F)(F)F.Cl.Cl
501.331
501.33
10mg
C22H21Cl2F3N4O2
UKMTYUXWLKQDNT-UHFFFAOYSA-N
5-methyl-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide;dihydrochloride
90488853
>99%
Videos