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RS 67506 hydrochloride, Tocris Bioscience™

5-HT4 partial agonist

Brand:  Tocris (Bio-Techne) 0990/10

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 10mg

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Product Code. 13448243

  • £111.72 / 10mg

Estimated Shipment date
from Supplier 17-12-2019

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Description

Description

A potent and selective 5-HT4 partial agonist, with a pKi of 8.8 at 5-HT4 sites in guinea pig striatum, but < 6.0 at several other receptors including 5-HT1A, 1D, 2A, 2C, D1, D2 and M1-3. It is active in vivo and has an intrinsic activity compared to 5-HT of 0.6.
Specifications

Chemical Identifiers

168986-61-6
454.407
rs 67506 hydrochloride, 1-4-amino-5-chloro-2-methoxyphenyl-3-1-2-methylsulphonylamino ethyl-4-piperidinyl-1-propanone hydrochloride, n-2-4-3-4-amino-5-chloro-2-methoxyphenyl-3-oxopropyl piperidin-1-yl ethyl methanesulfonamide hydrochloride, 1-4-amino-5-chloro-2-methoxyphenyl-3-1-2-methyl sulphonylamino ethyl-4-piperidinyl-1-propanone hydrochloride
N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]methanesulfonamide;hydrochloride
C18H29Cl2N3O4S
GFWKWEHKHLTRRF-UHFFFAOYSA-N
133075
COC1=CC(=C(C=C1C(=O)CCC2CCN(CC2)CCNS(=O)(=O)C)Cl)N.Cl

Specifications

10mg
168986-61-6
rs 67506 hydrochloride, 1-4-amino-5-chloro-2-methoxyphenyl-3-1-2-methylsulphonylamino ethyl-4-piperidinyl-1-propanone hydrochloride, n-2-4-3-4-amino-5-chloro-2-methoxyphenyl-3-oxopropyl piperidin-1-yl ethyl methanesulfonamide hydrochloride, 1-4-amino-5-chloro-2-methoxyphenyl-3-1-2-methyl sulphonylamino ethyl-4-piperidinyl-1-propanone hydrochloride
COC1=CC(=C(C=C1C(=O)CCC2CCN(CC2)CCNS(=O)(=O)C)Cl)N.Cl
454.407
454.41
RS 67506 hydrochloride
C18H29Cl2N3O4S
GFWKWEHKHLTRRF-UHFFFAOYSA-N
N-[2-[4-[3-(4-amino-5-chloro-2-methoxyphenyl)-3-oxopropyl]piperidin-1-yl]ethyl]methanesulfonamide;hydrochloride
133075
>98%
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