Remoxipride hydrochloride, Tocris Bioscience™

Selective D2-like antagonist

Brand:  Tocris (Bio-Techne) 091610

Product Code. 13458153

Description

Dopamine D2 receptor antagonist showing selectivity over D3 and D4 receptors (Ki values are ∽ 300, ∽ 1600, and ∽ 2800 nM for D2, D3 and D4 receptors respectively). Exhibits antipsychotic activity in vivo with no extrapyramidal side effects. 50-fold more potent than sulpiride in antagonising the effects of apomorphine in the rat.

Chemical Identifiers

• CAS: 73220-03-8
• Molecular Weight (g/mol): 407.733
• Synonym: (S)-(-)-3-Bromo-N-[(1-ethyl-2-pyrrolidinylmethyl]2, 6-dimethoxybenzamide hydrochloride

• Molecular Formula: C16H24BrClN2O3
• InChI Key: WCPXLMIPGMFZMY-MERQFXBCSA-N
• PubChem CID: 15565709

Specifications

• Chemical Name or Material: Remoxipride hydrochloride
• Purity Grade: >98%
• Synonym: (S)-(-)-3-Bromo-N-[(1-ethyl-2-pyrrolidinylmethyl]2, 6-dimethoxybenzamide hydrochloride
• SMILES: CCN1CCCC1CNC(=O)C2=C(C=CC(=C2OC)Br)OC.Cl
• Molecular Weight (g/mol): 407.733
• Quantity: 10mg

• CAS: 73220-03-8
• Molecular Formula: C16H24BrClN2O3
• InChI Key: WCPXLMIPGMFZMY-MERQFXBCSA-N
• IUPAC Name: 3-bromo-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]-2,6-dimethoxybenzamide;hydrochloride
• PubChem CID: 15565709
• Formula Weight: 407.73