L-798,106, Tocris Bioscience™

Potent and highly selective EP3 antagonist

Brand:  Tocris (Bio-Techne) 334210

Product Code. 13462844

Description

Potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2 respectively). Attenuates sulprostone-induced inhibition of EFS-evoked twitch and contractile responses in vivo.

Chemical Identifiers

• Chemical Name or Material: L-798, 106
• Molecular Formula: C₂₇H₂₂BrNO₄S
• Formula Weight: 536.44
• Synonym: N-[(5-Bromo-2-methoxyphenyl)sulfonyl]-3-[2-(2-naphthalenylmethyl)phenyl]-2-propenamide

Specifications

• Chemical Name or Material: L-798, 106
• Quantity: 10mg
• Molecular Formula: C₂₇H₂₂BrNO₄S
• Synonym: N-[(5-Bromo-2-methoxyphenyl)sulfonyl]-3-[2-(2-naphthalenylmethyl)phenyl]-2-propenamide

• CAS: 244101-02-8
• Purity Grade: >99%
• Formula Weight: 536.44