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HC 067047, Tocris Bioscience™

Potent and selective TRPV4 antagonist

Brand:  Tocris (Bio-Techne) 410050

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 50mg

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Product Code. 13454144

  • £635.04 / 50mg

Estimated Shipment date
from Supplier 30-03-2020

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Description

Description

Potent and selective TRPV4 antagonist. Reversibly inhibits currents through mouse, human and rat TRPV4 orthologs (IC50 values are 17, 48 and 133 nM respectively). Also inhibits the endogenous TRPV4-mediated response to 4α-PDH (IC50 = 22 nM). Selective for TRPV4 over TRPV1, TRPV2, TRPV3 and TRPM8 channels.
Specifications

Chemical Identifiers

883031-03-6
471.524
2-methyl-1-3-4-morpholinyl propyl-5-phenyl-n-3-trifluoromethyl phenyl-1h-pyrrole-3-carboxamide, d0b1qm, 2-methyl-1-3-morpholin-4-ylpropyl-5-phenyl-n-3-trifluoromethyl phenyl pyrrole-3-carboxamide, hc hplc, 2-methyl-1-3-morpholin-4-yl propyl-5-phenyl-n-3-trifluoromethyl phenyl-1h-pyrrole-3-carboxamide, n-3-trifluoromethyl phenyl-2-methyl-1-3-morpholinopropyl-5-phenyl-1h-pyrrole-3-carboxamide
2-methyl-1-(3-morpholin-4-ylpropyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide
C26H28F3N3O2
NCZYSQOTAYFTNM-UHFFFAOYSA-N
2742550
CC1=C(C=C(N1CCCN2CCOCC2)C3=CC=CC=C3)C(=O)NC4=CC=CC(=C4)C(F)(F)F

Specifications

50mg
883031-03-6
2-methyl-1-3-4-morpholinyl propyl-5-phenyl-n-3-trifluoromethyl phenyl-1h-pyrrole-3-carboxamide, d0b1qm, 2-methyl-1-3-morpholin-4-ylpropyl-5-phenyl-n-3-trifluoromethyl phenyl pyrrole-3-carboxamide, hc hplc, 2-methyl-1-3-morpholin-4-yl propyl-5-phenyl-n-3-trifluoromethyl phenyl-1h-pyrrole-3-carboxamide, n-3-trifluoromethyl phenyl-2-methyl-1-3-morpholinopropyl-5-phenyl-1h-pyrrole-3-carboxamide
CC1=C(C=C(N1CCCN2CCOCC2)C3=CC=CC=C3)C(=O)NC4=CC=CC(=C4)C(F)(F)F
471.524
471.51
HC 067047
C26H28F3N3O2
NCZYSQOTAYFTNM-UHFFFAOYSA-N
2-methyl-1-(3-morpholin-4-ylpropyl)-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide
2742550
>99%
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