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GR 127935 hydrochloride, Tocris Bioscience™

Potent and selective 5-HT1B and 5-HT1D antagonist

Brand:  Tocris (Bio-Techne) 1477/50

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 50mg

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Product Code. 13449333

  • £786.45 / 50mg

Estimated Shipment date
from Supplier 21-11-2019

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Description

Description

Potent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other receptor types. Centrally active following oral administration.
Specifications

Chemical Identifiers

148642-42-6
534.057
gr 127935 hydrochloride, gr127935 hydrochloride, gr 127935 hydrochloride hydrate, n-4-methoxy-3-4-methyl-1-piperazinyl phenyl-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl-1,1'-biphenyl-4-carboxamide hydrochloride, n-4-methoxy-3-4-methylpiperazin-1-yl phenyl-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl biphenyl-4-carboxamide hydrochloride, 4-2-methoxy-5-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl biphenyl-4-yl carbonyl amino phenyl-1-methylpiperazin-1-ium chloride
CHEBI:64111
CC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)N5CCN(CC5)C.Cl
C29H32ClN5O3
SRVVUYIJVBLEJI-UHFFFAOYSA-N
11497466
N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride

Specifications

50mg
148642-42-6
gr 127935 hydrochloride, gr127935 hydrochloride, gr 127935 hydrochloride hydrate, n-4-methoxy-3-4-methyl-1-piperazinyl phenyl-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl-1,1'-biphenyl-4-carboxamide hydrochloride, n-4-methoxy-3-4-methylpiperazin-1-yl phenyl-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl biphenyl-4-carboxamide hydrochloride, 4-2-methoxy-5-2'-methyl-4'-5-methyl-1,2,4-oxadiazol-3-yl biphenyl-4-yl carbonyl amino phenyl-1-methylpiperazin-1-ium chloride
CC1=C(C=CC(=C1)C2=NOC(=N2)C)C3=CC=C(C=C3)C(=O)NC4=CC(=C(C=C4)OC)N5CCN(CC5)C.Cl
534.057
CHEBI:64111
>99%
GR 127935 hydrochloride
C29H32ClN5O3
SRVVUYIJVBLEJI-UHFFFAOYSA-N
N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide;hydrochloride
11497466
534.06
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