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GR 113808, Tocris Bioscience™

Potent and selective 5-HT4 antagonist

Brand:  Tocris (Bio-Techne) 132250

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 50mg

 View more versions of this product

Product Code. 13439143

  • £689.43 / 50mg

Estimated Shipment date
from Supplier 20-11-2019

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Description

Description

Potent, selective 5-HT4 receptor antagonist (pKB = 9.43 in human colonic muscle, and Kd = 0.15 nM for binding to cloned human 5-HT4 receptors). Displays > 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors.
Specifications

Chemical Identifiers

144625-51-4
393.502
unii-zt350oyt3i, zt350oyt3i, 1-2-methylsulfonylamino ethyl-4-piperidinyl methyl 1-methyl-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 1-methyl-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, 1-2-methylsulfonyl amino ethyl piperidin-4-yl methyl 1-methyl-1h-indole-3-carboxylate, 1-2-methanesulfonamidoethyl piperidin-4-yl methyl 1-methylindole-3-carboxylate, 1-2-methylsulfonyl-amino ethyl-4-piperidinyl methyl 1-methyl-1h-indole-3-carboxylate, 1-methyl-1h-indole-3-carboxylic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, tocris-1322, lopac-g-5918
CHEBI:73380
CN1C=C(C2=CC=CC=C21)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C
C19H27N3O4S
MOZPSIXKYJUTKI-UHFFFAOYSA-N
119376
[1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 1-methylindole-3-carboxylate

Specifications

50mg
144625-51-4
unii-zt350oyt3i, zt350oyt3i, 1-2-methylsulfonylamino ethyl-4-piperidinyl methyl 1-methyl-1h-indole-3-carboxylate, 1h-indole-3-carboxylic acid, 1-methyl-, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, 1-2-methylsulfonyl amino ethyl piperidin-4-yl methyl 1-methyl-1h-indole-3-carboxylate, 1-2-methanesulfonamidoethyl piperidin-4-yl methyl 1-methylindole-3-carboxylate, 1-2-methylsulfonyl-amino ethyl-4-piperidinyl methyl 1-methyl-1h-indole-3-carboxylate, 1-methyl-1h-indole-3-carboxylic acid, 1-2-methylsulfonyl amino ethyl-4-piperidinyl methyl ester, tocris-1322, lopac-g-5918
CN1C=C(C2=CC=CC=C21)C(=O)OCC3CCN(CC3)CCNS(=O)(=O)C
393.502
CHEBI:73380
>98%
GR 113808
C19H27N3O4S
MOZPSIXKYJUTKI-UHFFFAOYSA-N
[1-[2-(methanesulfonamido)ethyl]piperidin-4-yl]methyl 1-methylindole-3-carboxylate
119376
393.5
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