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GP 1a, Tocris Bioscience™

CB2 receptor inverse agonist

Brand:  Tocris (Bio-Techne) 276410

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 10mg

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Product Code. 13440544

  • £163.68 / 10mg

Estimated Shipment
09-07-2019

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Description

Description

CB2 receptor inverse agonist (pEC50 = 7.1), shown in cAMP, GTPγS and β-arrestin recruitment assays. Demonstrates approximately 30-fold selectivity for CB2 receptors over CB1 receptors. Increases P-ERK1/2 expression in HL-60 cells in vitro.
Specifications

Chemical Identifiers

511532-96-0
441.356
gp 1a, n-piperidin-1-yl-1-2,4-dichlorophenyl-1,4-dihydro-6-methylindeno 1,2-c pyrazole-3-carboxamide, 6-methyl-1-2,4-dichlorophenyl-n-piperidin-1-yl-1,4-dihydroindeno 1,2-c pyrazole-3-carboxamide
1-(2,4-dichlorophenyl)-6-methyl-N-piperidin-1-yl-4H-indeno[1,2-c]pyrazole-3-carboxamide
C23H22Cl2N4O
FNOMTMVRTBHRET-UHFFFAOYSA-N
10252734
CC1=CC2=C(C=C1)C3=C(C2)C(=NN3C4=C(C=C(C=C4)Cl)Cl)C(=O)NN5CCCCC5

Specifications

GP 1a
511532-96-0
C23H22Cl2N4O
FNOMTMVRTBHRET-UHFFFAOYSA-N
1-(2,4-dichlorophenyl)-6-methyl-N-piperidin-1-yl-4H-indeno[1,2-c]pyrazole-3-carboxamide
10252734
10mg
>99%
gp 1a, n-piperidin-1-yl-1-2,4-dichlorophenyl-1,4-dihydro-6-methylindeno 1,2-c pyrazole-3-carboxamide, 6-methyl-1-2,4-dichlorophenyl-n-piperidin-1-yl-1,4-dihydroindeno 1,2-c pyrazole-3-carboxamide
CC1=CC2=C(C=C1)C3=C(C2)C(=NN3C4=C(C=C(C=C4)Cl)Cl)C(=O)NN5CCCCC5
441.356
441.35
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