Tocris Bioscience™ Efaroxan hydrochloride

alpha2 antagonist and I1, I3 ligand

Description

Potent, highly selective α2 adrenoceptor antagonist and imidazoline I1 receptor ligand (pKi values are 7.87, 7.42, 5.74, 7.28 and < 5 for α 2A, α2B, α2C, I1, and I2 receptors respectively). Promotes insulin secretion, at a site distinct from I1 or I2 (the putative I3 receptor) in vitro and in vivo.

Specifications

• Assay Percent Range: >99%
• Chemical Name or Material: 2-(2-Ethyl-2,3-dihydro-2-benzofuranyl)-4,5-dihydro-1H-imidazole hydrochloride
• CAS: 89197-00-2

For Research Use Only