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BRL 54443, Tocris™

Potent 5-ht1E/F agonist

Brand:  Tocris (Bio-Techne) 112910

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 10mg

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Product Code. 13488613

  • £127.00 / 10mg


Estimated Shipment
02-11-2017
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Description

Description

A potent 5-ht1E/1F receptor agonist (pEC50 values are 8.5 and 8.6 respectively). Displays > 30-fold selectivity over other 5-HT and dopamine receptors (pKi values are 8.7. 8.9, 7.2, 6.9, 7.2, 5.9, 7.0, 6.5, < 6, < 6, 6.3 and 6.2 for human 5-HT1E, 1F, 1A, 1B, 1D, 2A, 2B, 2C, 4, 7, D2 and D3 receptors respectively). Induces 5-HT2A receptor-mediated mouse aortic contraction in vitro (pEC50 = 6.52). Active in vivo.
Specifications

Chemical Identifiers

BRL 54443
C14H18N2O
5-Hydroxy-3-(1-methylpiperidin-4-yl)-1H-indole
>98%
230.31

Specifications

BRL 54443
57477-39-1
C14H18N2O
5-Hydroxy-3-(1-methylpiperidin-4-yl)-1H-indole
10mg
>98%
230.31