missing translation for 'onlineSavingsMsg'
Learn More

BRL 54443, Tocris Bioscience™

Potent 5-ht1E/F agonist

Brand:  Tocris (Bio-Techne) 112950

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 50mg

 View more versions of this product

Product Code. 13458623

  • £396.52 / 50mg


Estimated Shipment
27-11-2018
Add to basket

Description

Description

A potent 5-ht1E/1F receptor agonist (pEC50 values are 8.5 and 8.6 respectively). Displays > 30-fold selectivity over other 5-HT and dopamine receptors (pKi values are 8.7. 8.9, 7.2, 6.9, 7.2, 5.9, 7.0, 6.5, < 6, < 6, 6.3 and 6.2 for human 5-HT1E, 1F, 1A, 1B, 1D, 2A, 2B, 2C, 4, 7, D2 and D3 receptors respectively). Induces 5-HT2A receptor-mediated mouse aortic contraction in vitro (pEC50 = 6.52). Active in vivo.
Specifications

Chemical Identifiers

57477-39-1
230.311
3-1-methylpiperidin-4-yl-1h-indol-5-ol, unii-q2dh1chi0y, q2dh1chi0y, 1h-indol-5-ol, 3-1-methyl-4-piperidinyl, 5-hydroxy-3-1-methylpiperidin-4-yl-1h-indole, 3-1-methyl-4-piperidinyl-1h-indol-5-ol, tocris-1129, lopac-b-173, biomol-nt_000107, d0q5sl
3-(1-methylpiperidin-4-yl)-1H-indol-5-ol
C14H18N2O
WKNFADCGOAHBPG-UHFFFAOYSA-N
2438
CN1CCC(CC1)C2=CNC3=C2C=C(C=C3)O

Specifications

BRL 54443
57477-39-1
3-1-methylpiperidin-4-yl-1h-indol-5-ol, unii-q2dh1chi0y, q2dh1chi0y, 1h-indol-5-ol, 3-1-methyl-4-piperidinyl, 5-hydroxy-3-1-methylpiperidin-4-yl-1h-indole, 3-1-methyl-4-piperidinyl-1h-indol-5-ol, tocris-1129, lopac-b-173, biomol-nt_000107, d0q5sl
CN1CCC(CC1)C2=CNC3=C2C=C(C=C3)O
230.311
230.31
50mg
C14H18N2O
WKNFADCGOAHBPG-UHFFFAOYSA-N
3-(1-methylpiperidin-4-yl)-1H-indol-5-ol
2438
>98%
Videos