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AM 251, Tocris Bioscience™

Potent CB1 antagonist; also GPR55 agonist

Brand:  Tocris (Bio-Techne) 111750

Code : Z1

Additional Details : Weight : 0.01000kg

Quantity 50mg

 View more versions of this product

Product Code. 13428583

  • £643.86 / 50mg

Estimated Shipment date
from Supplier 27-03-2020

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Description

Description

Potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors. Also potent GPR55 agonist (EC50 = 39 nM) and μ-opioid receptor antagonist (Ki = 251 nM).

Fluorescent Form also available.

Specifications

Chemical Identifiers

183232-66-8
555.241
unii-3i4fa44mai, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-yl-1h-pyrazole-3-carboxamide, n-piperidin-1-yl-5-4-iodophenyl-1-2,4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide, 3i4fa44mai, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-ylpyrazole-3-carboxamide, n-piperidin-1-yl-5-4-iodophenyl-1-2, 4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-1-piperidinyl-1h-pyrazole-3-carboxamide, am 251 pharmaceutical, tocris-1117, d08yqt
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
C22H21Cl2IN4O
BUZAJRPLUGXRAB-UHFFFAOYSA-N
2125
CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I

Specifications

50mg
183232-66-8
unii-3i4fa44mai, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-yl-1h-pyrazole-3-carboxamide, n-piperidin-1-yl-5-4-iodophenyl-1-2,4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide, 3i4fa44mai, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-ylpyrazole-3-carboxamide, n-piperidin-1-yl-5-4-iodophenyl-1-2, 4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide, 1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-1-piperidinyl-1h-pyrazole-3-carboxamide, am 251 pharmaceutical, tocris-1117, d08yqt
CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I
555.241
555.24
AM 251
C22H21Cl2IN4O
BUZAJRPLUGXRAB-UHFFFAOYSA-N
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
2125
>99%
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